SCHEMBL8312894

SCHEMBL8312894

CCc1cccc(Nc2ncnc3cnc(SC)nc23)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.51
ABCG2 Q9UNQ0 1/20 0.46
SYK P43405 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
GRM4 Q14833 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994562 0.90 EGFR (0.50) EGFRABCG2SYK
SCHEMBL6992120 0.85 EGFR (0.70) EGFRMAPK1HTT
SCHEMBL8314131 0.84 EGFR (0.53) EGFRABCG2MAPK1HTT
SCHEMBL8313726 0.84 EGFR (0.59) EGFRHTT
SCHEMBL8317436 0.84 EGFR (0.69) EGFR
SCHEMBL6996346 0.83 EGFR (0.47) EGFRABCG2HTT
SCHEMBL8320191 0.83 EGFR (0.65) EGFRABCG2MAPK1HTT
SCHEMBL8314069 0.82 EGFR (0.57) EGFRABCG2HTT
SCHEMBL7000944 0.81 EGFR (0.53) EGFRABCG2SYK
SCHEMBL8317468 0.81 EGFR (0.57) EGFRABCG2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed