SCHEMBL8317468

SCHEMBL8317468

CSc1ncc2ncnc(Nc3cccc(C(F)(F)F)c3)c2n1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.57
ABCG2 Q9UNQ0 2/20 0.56
TSHR P16473 1/20 0.55
HTT P42858 1/20 0.55
BRAF P15056 1/20 0.49
TRPV1 Q8NER1 1/20 0.48
CD38 P28907 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314131 0.85 EGFR (0.53) EGFRABCG2HTT
SCHEMBL6996977 0.84 SYK (0.50) EGFRBRAF
SCHEMBL6992120 0.84 EGFR (0.70) EGFRHTT
SCHEMBL8313726 0.83 EGFR (0.59) EGFRHTT
SCHEMBL8317436 0.83 EGFR (0.69) EGFR
SCHEMBL8320191 0.82 EGFR (0.65) EGFRABCG2HTT
SCHEMBL6992546 0.81 EGFR (0.45) EGFRABCG2BRAF
SCHEMBL8312894 0.81 EGFR (0.51) EGFRABCG2HTT
SCHEMBL8314069 0.81 EGFR (0.57) EGFRABCG2HTT
SCHEMBL8318188 0.81 EGFR (0.55) EGFRABCG2TSHRHTTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed