SCHEMBL8312962

SCHEMBL8312962

C#Cc1cccc(Nc2ncnc3cnc(N4CCC(=O)CC4)nc23)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.48
GAK O14976 2/20 0.46
RIPK2 O43353 1/20 0.46
BUB1 O43683 1/20 0.46
STK10 O94804 1/20 0.46
CARS1 P49589 1/20 0.46
MAP3K1 Q13233 1/20 0.46
PIP4K2C Q8TBX8 1/20 0.46
SLK Q9H2G2 1/20 0.46
ERBB2 P04626 2/20 0.46
ERBB4 Q15303 1/20 0.46
BRAF P15056 7/20 0.45
FBP1 P09467 2/20 0.45
MAPT P10636 2/20 0.45
ALDH1A1 P00352 1/20 0.45
AURKA O14965 1/20 0.43
RPS6KB1 P23443 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314998 0.90 BRAF (0.51) EGFRGAKRIPK2BUB1STK10
SCHEMBL8318130 0.87 EGFR (0.54) EGFRGAKRIPK2BUB1STK10
SCHEMBL8314587 0.85 EGFR (0.60) EGFRBRAF
SCHEMBL8315732 0.85 EGFR (0.60) EGFR
SCHEMBL8319394 0.85 EGFR (0.50) EGFRERBB2BRAFMAPT
SCHEMBL8318621 0.82 ABCG2 (0.52) EGFRBRAF
SCHEMBL7574919 0.81 BRAF (0.45) EGFRGAKERBB2ERBB4BRAF
SCHEMBL8318461 0.80 EGFR (0.55) EGFRERBB2BRAFMAPT
SCHEMBL8314683 0.79 CSNK2A1 (0.55) EGFRGAKRIPK2BUB1STK10
SCHEMBL8320166 0.78 EGFR (0.67) EGFRERBB2ERBB4BRAFMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed