SCHEMBL8313110

SCHEMBL8313110

CC(C)(C)Cc1csc(-c2cc3cc(O)ccc3o2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
APP P05067 7/20 0.44
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
MIF P14174 1/20 0.38
PDE4D Q08499 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
CASP1 P29466 1/20 0.37
BRCA1 P38398 1/20 0.37
CASP7 P55210 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
LCK P06239 1/20 0.36
PTGES O14684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310416 0.84 ESR1 (0.42) ESR1ESR2APPPDE4DKDM4E
SCHEMBL8311404 0.83 ESR1 (0.48) ESR1ESR2APPPDE4DKDM4E
SCHEMBL27480747 0.81 ESR1 (0.43) ESR1ESR2APPKDM4EALDH1A1
SCHEMBL6600736 0.81 ESR1 (0.48) ESR1ESR2APPPDE4DKDM4E
SCHEMBL8315658 0.81 ALOX15 (0.43) ESR1ESR2APPMIFKDM4E
SCHEMBL8314204 0.80 KDM4E (0.39) ESR1ESR2APPKDM4EALDH1A1
SCHEMBL8316603 0.80 ALOX15 (0.42) ESR1ESR2APPMIFKDM4E
SCHEMBL8310912 0.79 MIF (0.54) ESR1ESR2APPMIFKDM4E
SCHEMBL8314199 0.78 KDM4E (0.38) ESR1ESR2APPKDM4EALDH1A1
SCHEMBL8310437 0.76 F2RL3 (0.35) APPCNR1CNR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
CN-1036589-C New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1997-12-03 CN disclosed
CN-1033088-C Thiazolylbenzofuran derivatives, processes for preparation thereof and pharmaceutical composition comprising same FUJISAWA PHARMACEUTICAL CO (JP) 1996-10-23 CN disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
CN-1074444-A New thiazolyl benzofuran derivative, its preparation method and contain the pharmaceutical composition of this derivative FUJISAWA PHARMACEUTICAL CO (JP) 1993-07-21 CN disclosed
CN-1070910-A New thiazolyl benzofuran derivative, its preparation method and contain the pharmaceutical composition of this derivative FUJISAWA PHARMACEUTICAL CO (JP) 1993-04-14 CN disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed