SCHEMBL8313156

SCHEMBL8313156

Cc1c(C#N)sc2nc(-c3ccc4c(c3)OCO4)nc(N3CCC(C)(N)CC3)c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
HSD17B10 Q99714 6/20 0.53
HPGD P15428 4/20 0.53
TSHR P16473 3/20 0.53
KDM4E B2RXH2 3/20 0.53
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
USP2 O75604 2/20 0.41
CYP2C19 P33261 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
KIT P10721 5/20 0.41
ALOX15 P16050 4/20 0.39
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
PIK3CG P48736 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 1/20 0.37
ADORA1 P30542 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2837286 0.87 ALDH1A1 (0.57) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL2834416 0.87 ALDH1A1 (0.57) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8311286 0.85 ALDH1A1 (0.64) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8306834 0.84 KDM4E (0.55) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8312062 0.83 KDM4E (0.61) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8312543 0.83 KDM4E (0.77) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8306844 0.81 ALDH1A1 (0.59) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8311877 0.81 KDM4E (0.58) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8306886 0.80 KDM4E (0.57) ALDH1A1HSD17B10HPGDTSHRKDM4E
SCHEMBL8313961 0.78 ALDH1A1 (0.52) ALDH1A1HSD17B10HPGDTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065391-A1 4-AMINOTHIENO[2,3-d]PYRIMIDINE-6-CARBONITRILE DERIVATIVES AS PDE7 INHIBITORS ALMIRALL PRODESFARMA S.A. (ES) 2004-08-05 WO disclosed