SCHEMBL8313158

SCHEMBL8313158

OCCCC(CO)(c1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
HIF1A Q16665 1/20 0.39
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
MIF P14174 1/20 0.37
KIF11 P52732 1/20 0.37
CCR1 P32246 3/20 0.34
CCR3 P51677 3/20 0.34
CYP19A1 P11511 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312683 0.93 KIF11 (0.47) BCL2MEN1KMT2ATSHRMAPK1
SCHEMBL5732977 0.88 TSHR (0.41) BCL2MEN1KMT2ATSHRMAPK1
SCHEMBL7462429 0.86 CCR1 (0.44) BCL2MEN1KMT2ATSHRMAPK1
SCHEMBL7830838 0.80 KIF11 (0.54) BCL2TSHRMIFKIF11CCR1
SCHEMBL8310962 0.79 CHRM3 (0.39) MEN1KMT2ATSHRESR1ESR2
SCHEMBL8314216 0.78 CHRM3 (0.38) TSHRMAPK1ESR1ESR2KIF11
SCHEMBL2009309 0.78 BCL2 (0.62) BCL2MEN1KMT2ATSHRMAPK1
SCHEMBL7825245 0.77 CCR3 (0.39) BCL2MEN1KMT2AMIFCCR1
SCHEMBL8310441 0.74 KCNN4 (0.42) MEN1KMT2AESR1ESR2KIF11
SCHEMBL10339814 0.71 TSHR (0.38) BCL2MEN1KMT2ATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679642-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-11-10 EP disclosed
US-5654296-A HORMONE INHIBITOR; NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-08-05 US disclosed
US-5607939-A CALCIUM ANTAGONIST, GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONIST AND MONOAMINEU UPTAKE INHIBITORS FOR CENTRAL NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-04 US disclosed
EP-0679642-A1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-02 EP disclosed