SCHEMBL8313667

SCHEMBL8313667

Cc1ccc2c(c1)C(N)NO2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.39
HTR2C P28335 4/20 0.36
HTR2B P41595 2/20 0.36
HTR1A P08908 1/20 0.36
SLC6A2 P23975 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
MAPT P10636 3/20 0.33
ALDH1A1 P00352 3/20 0.33
ADRA2A P08913 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR2A P28223 1/20 0.33
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
MMP12 P39900 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
TDP1 Q9NUW8 2/20 0.31
KMT2A Q03164 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14538282 0.85 ALDH1A1 (0.36) GAAHTR2CHTR2BHTR1ASLC6A2
SCHEMBL7920680 0.78 GAA (0.37) GAAHTR2CHTR2BHTR1ASLC6A2
SCHEMBL14748209 0.77 KDM1A (0.39) HTR2CHTR2BCHRNB2CHRNA4ALDH1A1
SCHEMBL7923004 0.67 ALDH1A1 (0.37) GAAHTR2CHTR2BSLC6A2CHRNB2
SCHEMBL10145621 0.65 HTR2C (0.46) GAAHTR2CHTR2BHTR1ASLC6A2
SCHEMBL16199826 0.65 ALDH1A1 (0.36) GAAHTR2CCHRNB2CHRNA4MAPT
SCHEMBL431417 0.63 ADRA2A (0.50) GAAHTR2CHTR2BHTR1ASLC6A2
SCHEMBL19756620 0.63 GAA (0.37) GAAHTR2CHTR2BHTR1ASLC6A2
Hydrochloric Acid SCHEMBL4809903 0.62 ADRA2A (0.49) GAAHTR2CHTR2BHTR1ASLC6A2
SCHEMBL9582603 0.62 CREBBP (0.42) GAAHTR2CHTR2BHTR1ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004083177-A2 LINEAR CHAIN SUBSTITUTED MONOCYCLIC AND BICYCLIC DERIVATIVES AS FACTOR XA INHIBITORS BRYSTOL-MYERS SQUIBB COMPANY (US) 2004-09-30 WO disclosed
WO-2004083174-A2 SULFONYL-AMIDINO CONTAINING AND TETRAHYDROPYRIMIDINO CONTAINING COMPOUNDS AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-09-30 WO disclosed