SCHEMBL8313758

SCHEMBL8313758

Cc1csc(-c2ccc[c]c2Cl)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.47
CYP3A4 P08684 2/20 0.42
CYP2E1 P05181 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2B6 P20813 1/20 0.42
GLA P06280 1/20 0.40
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ADORA2A P29274 3/20 0.38
ADRA1A P35348 1/20 0.36
TGFBR1 P36897 2/20 0.36
CYP19A1 P11511 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5324014 0.77 PDE10A (0.45) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL2096015 0.77 ALDH1A1 (0.59) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL11126054 0.74 PDE10A (0.49) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL8108203 0.72 CCR1 (0.50) CYP2A6TGFBR1
SCHEMBL5065334 0.72 PDPK1 (0.43) CYP2A6ADORA2AADRA1ACYP19A1RAB9A
SCHEMBL5584101 0.72 IDO1 (0.32) CYP2A6
SCHEMBL21091020 0.72 PDE10A (0.55) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL24181735 0.71 PDE10A (0.42) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL8198560 0.71 CYP3A4 (0.60) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL5536800 0.71 PDE10A (0.53) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901487-A1 NOVEL 2,3 DISUBSTITUTED-4(3H)-QUINAZOLINONES PFIZER INC. (US) 1999-03-17 EP disclosed
WO-1997043276-A1 NOVEL 2,3 DISUBSTITUTED-4(3H)-QUINAZOLINONES PFIZER INC. (US) 1997-11-20 WO disclosed