SCHEMBL8313783

SCHEMBL8313783

Cc1c([N+](=O)[O-])c2cnnc(OCc3ccccc3)c2n1CC(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGMT P16455 3/20 0.41
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PIN1 Q13526 2/20 0.39
CNR1 P21554 1/20 0.37
ACHE P22303 1/20 0.37
CNR2 P34972 1/20 0.37
LMNA P02545 4/20 0.36
ALDH1A1 P00352 5/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 1/20 0.34
HPGD P15428 2/20 0.33
ATM Q13315 2/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8940726 0.78 CYP1A2 (0.38) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
Fumaric Acid SCHEMBL8318500 0.78 CYP1A2 (0.38) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7485341 0.75 CYP1A2 (0.58) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7487573 0.70 CYP1A2 (0.57) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8314257 0.70 MAPT (0.47) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8314346 0.70 LMNA (0.51) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7480602 0.68 CYP1A2 (0.53) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7482125 0.68 CYP1A2 (0.53) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8311469 0.68 ALDH1A1 (0.37) CNR1ACHECNR2LMNAALDH1A1
SCHEMBL7482910 0.68 CYP1A2 (0.55) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609328-B1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-28 EP disclosed
US-5534515-A Pyrrolopyridazines having gastrointestinal protective effects BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-07-09 US disclosed
WO-1993008190-A1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1993-04-29 WO disclosed