SCHEMBL8314710

SCHEMBL8314710

CC(C)Oc1cc2cccc(N)c2cc1OC(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.50
MCHR1 Q99705 2/20 0.46
IRAK4 Q9NWZ3 5/20 0.45
ALDH1A1 P00352 4/20 0.41
HPGD P15428 3/20 0.41
CYP3A4 P08684 3/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KEAP1 Q14145 1/20 0.41
F2 P00734 1/20 0.39
PLG P00747 1/20 0.39
PLAU P00749 1/20 0.39
PLAT P00750 1/20 0.39
KLK1 P06870 1/20 0.39
PRSS1 P07477 1/20 0.39
MAPT P10636 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
POLB P06746 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315056 0.94 TLR8 (0.45) TLR8MCHR1IRAK4ALDH1A1HPGD
SCHEMBL19612294 0.80 CYP1A2 (0.46) TLR8MCHR1IRAK4ALDH1A1HPGD
SCHEMBL426014 0.79 ALDH1A1 (0.48) TLR8MCHR1ALDH1A1HPGDCYP3A4
SCHEMBL16606236 0.76 IRAK4 (0.61) TLR8MCHR1IRAK4ALDH1A1HPGD
SCHEMBL13865030 0.76 TLR8 (0.50) TLR8MCHR1IRAK4ALDH1A1HPGD
SCHEMBL28770352 0.76 ALDH1A1 (0.52) TLR8MCHR1IRAK4ALDH1A1HPGD
SCHEMBL5545202 0.73 ALDH1A1 (0.62) ALDH1A1HPGDCYP3A4TSHRHSD17B10
SCHEMBL29351158 0.73 ALDH1A1 (0.62) ALDH1A1HPGDCYP3A4TSHRHSD17B10
SCHEMBL2891381 0.71 ALDH1A1 (0.59) ALDH1A1HPGDCYP3A4TSHRHSD17B10
SCHEMBL29704534 0.71 ALDH1A1 (0.59) ALDH1A1HPGDCYP3A4TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487930-B1 Benzo[C]phenanthridinium derivatives NIPPON KAYAKU KK (JP) 1999-03-24 EP disclosed
US-5747502-A ANTITUMOR AGENTS, ANTIGROWTH AGENTS AND ANTICARCINOGENIC AGENTS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1998-05-05 US disclosed
EP-0487930-A1 Process for preparing benzo[C]phenanthridinium derivatives, and novel compounds prepared by said process NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-06-03 EP disclosed