SCHEMBL8314741

SCHEMBL8314741

O=C(O)CN(OCc1ccc(C(=O)O)cc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 8/20 0.49
RXRB P28702 7/20 0.49
RXRG P48443 5/20 0.49
HPGD P15428 1/20 0.49
NR4A2 P43354 3/20 0.47
NR4A1 P22736 1/20 0.47
NR4A3 Q92570 1/20 0.47
SRD5A2 P31213 2/20 0.44
PTGER1 P34995 1/20 0.44
PTGER4 P35408 1/20 0.44
PTGER3 P43115 1/20 0.44
PTGER2 P43116 1/20 0.44
PLA2G4B P0C869 1/20 0.42
ALDH1A1 P00352 1/20 0.42
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370663 0.89 ALDH1A1 (0.43) HPGDALDH1A1NPC1RAB9A
SCHEMBL8310205 0.74 ALDH1A1 (0.50) HPGDALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL27576865 0.74 ALDH1A1 (0.44) ALDH1A1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL11953861 0.73 ALDH1A1 (0.51) RXRARXRBRXRGHPGDNR4A2
SCHEMBL11133454 0.73 HTT (0.45) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL27832128 0.71 NR4A1 (0.67) RXRARXRBRXRGHPGDNR4A2
SCHEMBL1287366 0.70 SMN1; SMN2 (0.41) ALDH1A1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL7587208 0.70 ALDH1A1 (0.47) NR4A2NR4A1NR4A3ALDH1A1NPC1
SCHEMBL5089520 0.70 ALDH1A1 (0.42) HPGDALDH1A1NPC1POLBRAB9A
SCHEMBL8021970 0.70 ALDH1A1 (0.42) HPGDALDH1A1NPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934262-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-08-11 EP disclosed
WO-1998017639-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1998-04-30 WO disclosed