SCHEMBL8314824

SCHEMBL8314824

N#CCc1ccccc1COc1ccc2oc(-c3nc(-c4cccs4)cs3)cc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.42
MEN1 O00255 7/20 0.42
KMT2A Q03164 7/20 0.42
KDM4E B2RXH2 5/20 0.42
TDP1 Q9NUW8 3/20 0.42
POLB P06746 2/20 0.42
RAB9A P51151 6/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
HPGD P15428 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
CYP19A1 P11511 2/20 0.37
ALDH1A1 P00352 4/20 0.37
SREBF2 Q12772 1/20 0.35
MAOB P27338 1/20 0.34
NPC1 O15118 5/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
HSD17B10 Q99714 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310727 0.88 MAPT (0.44) MAPTMEN1KMT2AKDM4ETDP1
SCHEMBL8311847 0.88 KMT2A (0.39) MAPTMEN1KMT2AKDM4ETDP1
SCHEMBL8314218 0.86 CYP19A1 (0.41) MAPTMEN1KMT2AKDM4ETDP1
SCHEMBL8312884 0.85 MAPT (0.47) MAPTMEN1KMT2AKDM4ETDP1
SCHEMBL8310220 0.84 KDM4E (0.43) MAPTMEN1KMT2AKDM4ERAB9A
SCHEMBL8311876 0.83 FFAR4 (0.37) MAPTMEN1KMT2AKDM4ERAB9A
SCHEMBL8310631 0.82 F2RL3 (0.35) MAPTMEN1KMT2AKDM4ETDP1
SCHEMBL8310491 0.82 F2RL3 (0.33) MAPTMEN1KMT2AKDM4ECYP19A1
SCHEMBL8311729 0.82 F2RL3 (0.35) MAPTMEN1KMT2AKDM4ERAB9A
SCHEMBL8312101 0.81 MAPT (0.38) MAPTMEN1KMT2AKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed