SCHEMBL8314947

SCHEMBL8314947

Cc1cc2c(cc1Br)C(O)(c1ccccn1)CC(C)(C)CO2

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.37
SCN9A Q15858 2/20 0.36
GAA P10253 2/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
NFKB1 P19838 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314123 0.96 SLC6A2 (0.37) SLC6A2SCN9AGAALMNA
SCHEMBL8316835 0.85 SLC6A2 (0.39) SLC6A2GAANPC1MAPTNFKB1
SCHEMBL8310390 0.84 SLC6A2 (0.36) SLC6A2NPC1RAB9A
SCHEMBL8311974 0.84 BACE1 (0.37) SLC6A2MAPT
SCHEMBL8313558 0.84 SLC6A2 (0.38) SLC6A2SCN9A
SCHEMBL8316027 0.83 SCN9A (0.40) SLC6A2SCN9A
SCHEMBL8311725 0.81 SLC6A2 (0.36) SLC6A2
SCHEMBL8310494 0.81 SCN9A (0.38) SLC6A2SCN9ANPC1MAPTRAB9A
SCHEMBL8310708 0.81 SLC6A2 (0.40) SLC6A2
SCHEMBL8311266 0.81 SLC6A2 (0.37) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed