SCHEMBL8310708

SCHEMBL8310708

CC1(C)COc2ccccc2C(O)(c2ccccn2)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.40
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
PDK2 Q15119 2/20 0.32
KIF11 P52732 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
NR3C1 P04150 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311266 0.86 SLC6A2 (0.37) SLC6A2PDK2KIF11
SCHEMBL8316835 0.86 SLC6A2 (0.39) SLC6A2PDK2OPRM1OPRL1CYP1A2
SCHEMBL8311974 0.85 BACE1 (0.37) SLC6A2KMT2ASMN1; SMN2
SCHEMBL8313637 0.85 SLC6A2 (0.36) SLC6A2KMT2ANR3C1
SCHEMBL8310390 0.85 SLC6A2 (0.36) SLC6A2NR3C1
SCHEMBL8313558 0.85 SLC6A2 (0.38) SLC6A2CHRM2CHRM4CHRM5CHRM1
SCHEMBL8314119 0.84 HTR2B (0.38) SLC6A2PDK2KMT2AHTR1ASMN1; SMN2
SCHEMBL8316027 0.84 SCN9A (0.40) SLC6A2CHRM2CHRM4CHRM5CHRM1
SCHEMBL8313905 0.83 PDK2 (0.35) SLC6A2PDK2KMT2ANR3C1HPGD
SCHEMBL8314935 0.83 SCN9A (0.38) SLC6A2PDK2KMT2AHTR1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
EP-0626954-A1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GmbH (DE) 1994-12-07 EP disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed