SCHEMBL8313558

SCHEMBL8313558

CC1(C)COc2cc(Cl)c(Cl)cc2C(O)(c2ccccn2)C1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.38
NR3C1 P04150 1/20 0.33
AKR1B1 P15121 1/20 0.33
OPRM1 P35372 5/20 0.32
OPRL1 P41146 4/20 0.32
LDHA P00338 1/20 0.32
LDHB P07195 1/20 0.32
MAP3K14 Q99558 1/20 0.32
TAAR1 Q96RJ0 1/20 0.31
TRPV3 Q8NET8 1/20 0.31
SCN9A Q15858 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM4 P08173 1/20 0.30
CHRM5 P08912 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30
SLC6A9 P48067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315996 0.91 SLC6A2 (0.35) SLC6A2NR3C1AKR1B1OPRM1TRPV3
SCHEMBL8313637 0.88 SLC6A2 (0.36) SLC6A2NR3C1MAP3K14SLC6A9
SCHEMBL8316027 0.87 SCN9A (0.40) SLC6A2NR3C1OPRM1OPRL1TRPV3
SCHEMBL8311725 0.85 SLC6A2 (0.36) SLC6A2NR3C1
SCHEMBL8310494 0.85 SCN9A (0.38) SLC6A2SCN9A
SCHEMBL8310708 0.85 SLC6A2 (0.40) SLC6A2NR3C1OPRM1OPRL1TAAR1
SCHEMBL8311266 0.84 SLC6A2 (0.37) SLC6A2AKR1B1TRPV3
SCHEMBL8316835 0.84 SLC6A2 (0.39) SLC6A2NR3C1OPRM1OPRL1
SCHEMBL8314947 0.84 SLC6A2 (0.37) SLC6A2SCN9A
SCHEMBL8314123 0.84 SLC6A2 (0.37) SLC6A2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed