SCHEMBL8314951

SCHEMBL8314951

Fc1cc(F)cc(Nc2ncnc3cnc(NC4CC4)nc23)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.58
ERBB2 P04626 1/20 0.58
HPGD P15428 1/20 0.58
HTT P42858 1/20 0.58
CSNK2A1 P68400 3/20 0.54
BRAF P15056 4/20 0.48
CSNK2A2 P19784 2/20 0.45
CSNK2B P67870 2/20 0.45
MAP4K4 O95819 1/20 0.42
CTSV O60911 1/20 0.41
PLAT P00750 1/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSH P09668 1/20 0.41
CTSS P25774 1/20 0.41
CASP14 P31944 1/20 0.41
CTSK P43235 1/20 0.41
CASP4 P49662 1/20 0.41
CASP5 P51878 1/20 0.41
CASP6 P55212 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317928 0.89 EGFR (0.60) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8315463 0.88 EGFR (0.61) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8319410 0.86 EGFR (0.57) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317453 0.85 EGFR (0.69) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317815 0.85 EGFR (0.53) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8320277 0.84 CSNK2A1 (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8320282 0.84 CSNK2A1 (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8316261 0.82 EGFR (0.68) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314263 0.82 EGFR (0.84) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317972 0.81 BRAF (0.59) EGFRERBB2HPGDHTTCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed