SCHEMBL8317815

SCHEMBL8317815

FC(F)(F)c1cc(Nc2ncnc3cnc(NC4CC4)nc23)cc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.53
ERBB2 P04626 1/20 0.53
HPGD P15428 1/20 0.53
HTT P42858 1/20 0.53
CSNK2A1 P68400 2/20 0.47
CSNK2A2 P19784 1/20 0.47
CSNK2B P67870 1/20 0.47
CSNK2A3 Q8NEV1 1/20 0.47
CTSC P53634 1/20 0.47
BRAF P15056 4/20 0.46
ULK1 O75385 5/20 0.43
IRAK4 Q9NWZ3 1/20 0.43
AXL P30530 1/20 0.42
TYRO3 Q06418 1/20 0.42
MERTK Q12866 1/20 0.42
ULK2 Q8IYT8 1/20 0.42
PAK1 Q13153 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318987 0.89 CTSC (0.61) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314951 0.85 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8319410 0.83 EGFR (0.57) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314154 0.82 BRAF (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8316151 0.82 EGFR (0.64) EGFRERBB2HPGDHTTBRAF
SCHEMBL8315463 0.80 EGFR (0.61) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8315669 0.80 EGFR (0.56) EGFRERBB2HPGDHTTBRAF
SCHEMBL8317453 0.80 EGFR (0.69) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317928 0.79 EGFR (0.60) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314012 0.78 SYK (0.53) EGFRERBB2HPGDHTTCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed