SCHEMBL8315809

SCHEMBL8315809

CC1(C)C=C(c2cccc[n+]2[O-])c2ccc(C#N)cc2OC1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 2/20 0.60
ABCC8 Q09428 2/20 0.60
KCNJ11 Q14654 2/20 0.60
KCNJ8 Q15842 2/20 0.60
OPRD1 P41143 1/20 0.33
DAO P14920 1/20 0.32
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311739 0.91 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8OPRD1
SCHEMBL8314283 0.83 ABCC9 (0.42) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8312379 0.83 ABCC9 (0.45) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8315817 0.83 ABCC9 (0.45) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8316384 0.82 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8OPRD1
SCHEMBL8310653 0.82 ABCC9 (0.44) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8313597 0.80 ABCC9 (0.50) ABCC9ABCC8KCNJ11KCNJ8OPRD1
SCHEMBL8310360 0.79 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8312666 0.79 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL6369348 0.77 ABCC9 (0.62) ABCC9ABCC8KCNJ11KCNJ8OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP claimed
EP-0626954-A1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GmbH (DE) 1994-12-07 EP claimed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO claimed
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed