SCHEMBL8315840

SCHEMBL8315840

CC1(C)COc2ccc(OC(F)(F)F)cc2C(O)(c2cccc[n+]2[O-])C1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.33
CTSD P07339 1/20 0.33
CCR6 P51684 3/20 0.31
KCNH2 Q12809 2/20 0.31
DRD4 P21917 1/20 0.31
PRCP P42785 1/20 0.31
P2RY1 P47900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315522 0.88 BACE1 (0.33) BACE1CTSDDRD4
SCHEMBL8315199 0.85 ABCC9 (0.33)
SCHEMBL8310355 0.84 AKR1B1 (0.34)
SCHEMBL8313650 0.82 PDK2 (0.32)
SCHEMBL8315276 0.81 BACE1 (0.33) BACE1
SCHEMBL8315596 0.81 MAP3K14 (0.34)
SCHEMBL8314858 0.81
SCHEMBL8313605 0.81 HTR2B (0.35) BACE1CTSD
SCHEMBL8311155 0.79 AKR1B1 (0.32)
SCHEMBL8314357 0.79 ALDH1A1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed