SCHEMBL8315849

SCHEMBL8315849

CC(C)Oc1cccc(CC(=O)N(C)CC(CC[N+]23CCC(CC2)CC3)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.43
CCR5 P51681 2/20 0.42
TACR2 P21452 10/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8953619 0.99 TACR1 (0.42) TACR1CCR5TACR2
SCHEMBL8316040 0.87 TACR1 (0.40) TACR1CCR5TACR2
SCHEMBL8314434 0.87 CCR5 (0.48) TACR1CCR5TACR2
Hydrochloric Acid SCHEMBL8953696 0.86 TACR1 (0.39) TACR1CCR5TACR2
Hydrochloric Acid SCHEMBL8636368 0.86 CCR5 (0.47) TACR1CCR5TACR2
SCHEMBL8119238 0.84 CCR5 (0.42) TACR1CCR5TACR2
SCHEMBL8364651 0.84 CCR5 (0.46) TACR1CCR5TACR2
Iodide SCHEMBL8125149 0.84 CCR5 (0.42) TACR1CCR5TACR2
SCHEMBL8126875 0.80 CCR5 (0.42) TACR1CCR5TACR2
SCHEMBL9679089 0.79 TACR2 (0.53) TACR1CCR5TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591040-B1 Quaternary basic amides as tachykinines antagonists SANOFI SA (FR) 1999-02-03 EP disclosed
EP-0591040-A1 Quaternary basic amides as tachykinines antagonists SANOFI (FR) 1994-04-06 EP disclosed