SCHEMBL8316040

SCHEMBL8316040

CC(=O)OCCN(CC(CC[N+]12CCC(CC1)CC2)c1ccc(Cl)c(Cl)c1)C(=O)Cc1cccc(OC(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.40
TACR2 P21452 6/20 0.39
CCR5 P51681 2/20 0.32
MCHR1 Q99705 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
FDFT1 P37268 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8953696 0.99 TACR1 (0.39) TACR1TACR2CCR5MCHR1SLC6A2
SCHEMBL8315849 0.87 TACR1 (0.43) TACR1TACR2CCR5
SCHEMBL8315878 0.87 TACR1 (0.39) TACR1TACR2CCR5FDFT1
Hydrochloric Acid SCHEMBL8953619 0.86 TACR1 (0.42) TACR1TACR2CCR5
SCHEMBL8314053 0.83 TACR1 (0.37) TACR1TACR2CCR5FDFT1
Hydrochloric Acid SCHEMBL8953818 0.80 CCR5 (0.37) TACR1TACR2CCR5
SCHEMBL8592468 0.79 TACR1 (0.40) TACR1TACR2CCR5FDFT1
SCHEMBL8592517 0.76 TACR1 (0.38) TACR1TACR2CCR5FDFT1
SCHEMBL8591139 0.75 TACR1 (0.42) TACR1TACR2CCR5SLC6A3
SCHEMBL8314434 0.75 CCR5 (0.48) TACR1TACR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591040-B1 Quaternary basic amides as tachykinines antagonists SANOFI SA (FR) 1999-02-03 EP disclosed
EP-0591040-A1 Quaternary basic amides as tachykinines antagonists SANOFI (FR) 1994-04-06 EP disclosed