SCHEMBL8315855

SCHEMBL8315855

CC(C)(C)c1csc(-c2cc3cc(CSc4ccccc4C(=O)O)ccc3o2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.48
PRNP P04156 1/20 0.48
PTPRG P23470 1/20 0.43
CYP26A1 O43174 1/20 0.39
CYP26B1 Q9NR63 1/20 0.39
PTPRF P10586 4/20 0.37
PTPN2 P17706 4/20 0.37
PTPN1 P18031 4/20 0.37
FFAR1 O14842 1/20 0.36
KMT2A Q03164 5/20 0.36
MEN1 O00255 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314759 0.86 CYP26A1 (0.34) RAB9APRNPCYP26A1CYP26B1FFAR1
SCHEMBL8316064 0.85 FFAR1 (0.42) RAB9APRNPCYP26A1CYP26B1PTPRF
SCHEMBL8316475 0.85 CYP26A1 (0.33) RAB9ACYP26A1CYP26B1FFAR1KMT2A
SCHEMBL9400022 0.84 PTPRG (0.40) RAB9APRNPPTPRGCYP26A1CYP26B1
SCHEMBL8314615 0.82 MAPT (0.33) RAB9ACYP26A1CYP26B1KMT2AMEN1
SCHEMBL8310203 0.78
SCHEMBL8316517 0.78 BCL2 (0.43) RAB9AKMT2AMEN1ALDH1A1CA12
SCHEMBL8311225 0.78 CYP26A1 (0.42) RAB9ACYP26A1CYP26B1FFAR1KMT2A
SCHEMBL8310165 0.78 FFAR1 (0.56) RAB9ACYP26A1CYP26B1FFAR1KMT2A
SCHEMBL8311016 0.78 CYP26B1 (0.42) RAB9ACYP26A1CYP26B1FFAR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed