SCHEMBL8315864

SCHEMBL8315864

CC(C)Nc1ncc2ncnc(Nc3cccc(Cl)c3)c2n1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.58
CSNK2A2 P19784 1/20 0.57
CSNK2B P67870 1/20 0.57
CSNK2A1 P68400 1/20 0.57
CCNB2 O95067 2/20 0.52
CDK1 P06493 2/20 0.52
CCNB1 P14635 2/20 0.52
CCNB3 Q8WWL7 2/20 0.52
FADS1 O60427 1/20 0.51
LCK P06239 1/20 0.50
ERBB2 P04626 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313472 0.88 EGFR (0.53) EGFRCSNK2A2CSNK2BCSNK2A1CCNB2
SCHEMBL8318451 0.87 EGFR (0.77) EGFR
SCHEMBL8317099 0.86 EGFR (0.77) EGFR
SCHEMBL8315646 0.86 EGFR (0.58) EGFRLCK
SCHEMBL8314176 0.86 EGFR (0.53) EGFRCSNK2A2CSNK2BCSNK2A1FADS1
SCHEMBL8314039 0.85 EGFR (0.52) EGFRCSNK2A2CSNK2BCSNK2A1ERBB2
SCHEMBL6993701 0.84 EGFR (0.64) EGFRERBB2
SCHEMBL8316788 0.84 EGFR (0.58) EGFRFADS1LCKERBB2
SCHEMBL8318849 0.84 EGFR (0.55) EGFRCSNK2A1LCKERBB2
SCHEMBL8314074 0.82 ABCG2 (0.55) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed