SCHEMBL8315869

SCHEMBL8315869

CCOC(=O)c1ccccc1C=Cc1ccc2oc(-c3nc(C(C)(C)C)cs3)cc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
CYP26B1 Q9NR63 1/20 0.37
MAOB P27338 2/20 0.37
MAPT P10636 3/20 0.36
TP53 P04637 1/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
MAOA P21397 1/20 0.36
DHODH Q02127 2/20 0.35
CYP3A4 P08684 1/20 0.35
RAB9A P51151 2/20 0.35
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA7 P43166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315866 1.00 JAK2 (0.39) JAK2JAK3CYP26B1MAOBMAPT
SCHEMBL8314166 0.80 CA12 (0.41) JAK2JAK3CYP26B1MAOBMAPT
SCHEMBL6598801 0.77 CYP26B1 (0.58) CYP26B1MAPTCYP3A4CA12CA2
SCHEMBL6598831 0.75 L3MBTL1 (0.37) JAK2JAK3MAPTCASP3SENP8
SCHEMBL6599382 0.75 JAK2 (0.35) JAK2JAK3MAOBMAPTTP53
SCHEMBL6599461 0.75 FFAR1 (0.41) CYP26B1MAPTRAB9ACA12CA2
SCHEMBL8553966 0.74 JAK2 (0.36) JAK2JAK3MAOBMAPTTP53
SCHEMBL6600992 0.74 CHRM2 (0.41) CYP26B1MAOBMAPTRAB9AKDM4E
SCHEMBL6599628 0.74 RAB9A (0.42) MAPTRAB9ACA12CA2CA3
SCHEMBL8311230 0.73 CA12 (0.37) CYP26B1MAPTTP53CASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed