SCHEMBL8316093

SCHEMBL8316093

CC1(CF)C=Cc2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
XDH P47989 1/20 0.47
CA9 Q16790 2/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
TLR3 O15455 2/20 0.44
HIF1A Q16665 6/20 0.44
EPAS1 Q99814 5/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
GFER P55789 1/20 0.43
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
AKR1B1 P15121 1/20 0.38
ALDH1A1 P00352 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976994 0.87 PTGS1 (0.62) PTGS1PTGS2XDHCA9CA12
SCHEMBL6987818 0.84 TLR3 (0.46) PTGS1PTGS2XDHCA9CA12
SCHEMBL3193294 0.81 TLR3 (0.59) CA9CA12CA1TLR3HIF1A
SCHEMBL8315997 0.78 CA9 (0.49) PTGS1PTGS2XDHCA9CA12
SCHEMBL6948888 0.77 MAPT (0.47) PTGS1PTGS2XDHCA9CA12
SCHEMBL27330130 0.76 CA9 (0.50) CA9CA12CA1TLR3HIF1A
SCHEMBL8535288 0.76 TLR3 (0.46) PTGS1PTGS2XDHCA9CA12
SCHEMBL9531520 0.74 HIF1A (0.46) PTGS1PTGS2XDHTLR3HIF1A
SCHEMBL8134327 0.74 KMT2A (0.43) CA9CA12CA1TLR3HIF1A
SCHEMBL3258594 0.73 CA9 (0.44) PTGS1PTGS2XDHCA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632033-B1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1999-04-07 EP disclosed
US-5646308-A POTASSIUM CHANNEL ACTIVATORS USED AS ANTIASTHMATICS, ANTIEPILEPTICS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1997-07-08 US disclosed
EP-0632033-A1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-01-04 EP disclosed