SCHEMBL8316366

SCHEMBL8316366

CO[C@H]1CC[C@H](Nc2ncc3ncnc(Nc4ccc(Cl)c(Cl)c4)c3n2)CC1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.63
ERBB2 P04626 7/20 0.63
HPGD P15428 1/20 0.63
HTT P42858 1/20 0.63
EPHA2 P29317 7/20 0.46
KDR P35968 7/20 0.46
EPHB4 P54760 7/20 0.46
BCL6 P41182 2/20 0.46
BRAF P15056 1/20 0.45
FLT1 P17948 2/20 0.43
MAPK3 P27361 1/20 0.43
CSNK2A1 P68400 1/20 0.43
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316373 1.00 EGFR (0.63) EGFRERBB2HPGDHTTEPHA2
SCHEMBL8316240 0.92 EGFR (0.69) EGFRERBB2HPGDHTTEPHA2
SCHEMBL8318083 0.92 EGFR (0.76) EGFRERBB2HPGDHTTKDR
SCHEMBL8318086 0.92 EGFR (0.76) EGFRERBB2HPGDHTTKDR
SCHEMBL8319178 0.88 EGFR (0.57) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319173 0.88 EGFR (0.57) EGFRERBB2HPGDHTTBRAF
SCHEMBL8315620 0.87 EGFR (0.64) EGFRERBB2HPGDHTTBCL6
SCHEMBL8313702 0.87 EGFR (0.64) EGFRERBB2HPGDHTTBCL6
SCHEMBL8315344 0.87 EGFR (0.64) EGFRERBB2HPGDHTTBCL6
SCHEMBL8315348 0.87 EGFR (0.64) EGFRERBB2HPGDHTTBCL6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed