SCHEMBL8316997

SCHEMBL8316997

O=C1C(c2c[nH]c3cc(F)ccc23)=C(c2c[nH]c3cc(F)ccc23)C(=O)N1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.53
TACR1 P25103 1/20 0.46
HTR6 P50406 2/20 0.44
ATM Q13315 1/20 0.43
SSTR1 P30872 1/20 0.43
SSTR2 P30874 1/20 0.43
SSTR4 P31391 1/20 0.43
SSTR3 P32745 1/20 0.43
SSTR5 P35346 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CCNE2 O96020 1/20 0.41
PRKACA P17612 1/20 0.41
PRKACG P22612 1/20 0.41
PRKACB P22694 1/20 0.41
CCNE1 P24864 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9000991 0.82 CDK4 (0.44) HTR6CDK4CCND1CCNE2PRKACA
SCHEMBL9375258 0.80 SIRT2 (0.49) SIRT2TACR1HTR6ATMSSTR1
SCHEMBL8314260 0.79 SIRT2 (0.69) SIRT2TACR1CDK4CCND1CCNE2
SCHEMBL8315890 0.77 NQO1 (0.53) TACR1HTR6ATMSMN1; SMN2CA9
SCHEMBL8313886 0.75 PRKACA (0.61) SIRT2TACR1SMN1; SMN2CDK4CCND1
SCHEMBL18669003 0.72 CA9 (0.61) ATMSMN1; SMN2CA9CA1CA2
SCHEMBL8317402 0.71 SIRT2 (0.63) SIRT2HTR6CDK4CCND1CCNE2
SCHEMBL7193605 0.70 SIRT2 (1.00) SIRT2TACR1CDK4CCND1CCNE2
SCHEMBL8317087 0.70 ATM (0.58) ATMSMN1; SMN2CA9CA1CA2
SCHEMBL8316640 0.67 SIRT2 (0.68) SIRT2SMN1; SMN2CA9CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP disclosed
US-5547976-A VIRICIDES, HERPES VIRUS, CYTOMEGALOVIRUS; CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1996-08-20 US disclosed
EP-0630242-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1994-12-28 EP disclosed
WO-1993018766-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO disclosed