SCHEMBL8316640

SCHEMBL8316640

O=C1C(c2c[nH]c3ccccc23)=C(c2c[nH]c3ccccc23)C(=O)N1Cc1cccc([N+](=O)[O-])c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.68
ALDH1A1 P00352 3/20 0.54
HPGD P15428 1/20 0.54
HTT P42858 1/20 0.54
BCL2 P10415 1/20 0.53
SIRT1 Q96EB6 1/20 0.48
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
GAA P10253 1/20 0.47
GFER P55789 1/20 0.47
CA12 O43570 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
PKM P14618 1/20 0.46
PKLR P30613 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
ELANE P08246 1/20 0.44
CASP1 P29466 1/20 0.44
CASP3 P42574 1/20 0.44
CASP4 P49662 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7193605 0.82 SIRT2 (1.00) SIRT2HTTSIRT1KMT2AMEN1
SCHEMBL31687464 0.78 ALDH1A1 (0.73) ALDH1A1HPGDHTTKMT2AMEN1
SCHEMBL2049541 0.78 ALDH1A1 (0.73) ALDH1A1HPGDHTTKMT2AMEN1
SCHEMBL28006388 0.76 RAB9A (0.54) SIRT2ALDH1A1HPGDHTTBCL2
SCHEMBL8318378 0.76 NQO1 (0.68) ALDH1A1HPGDHTTKMT2AMEN1
SCHEMBL8322554 0.74 SIRT2 (0.74) SIRT2SIRT1KMT2AMEN1GAA
SCHEMBL23649349 0.74 ELANE (0.60) ALDH1A1BCL2KMT2AMEN1GAA
SCHEMBL29824887 0.74 ELANE (0.60) ALDH1A1BCL2KMT2AMEN1GAA
SCHEMBL8314260 0.74 SIRT2 (0.69) SIRT2SIRT1
SCHEMBL2952856 0.73 PKM (0.64) ALDH1A1BCL2KMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP disclosed
US-5547976-A VIRICIDES, HERPES VIRUS, CYTOMEGALOVIRUS; CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1996-08-20 US disclosed
EP-0630242-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1994-12-28 EP disclosed
WO-1993018766-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO disclosed