SCHEMBL8315890

SCHEMBL8315890

O=C1c2c(c3c4ccc(F)cc4[nH]c3c3[nH]c4cc(F)ccc4c23)C(=O)N1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.53
CDK4 P11802 4/20 0.47
CCND1 P24385 4/20 0.47
CCNE2 O96020 2/20 0.46
CCNE1 P24864 2/20 0.46
CDK2 P24941 2/20 0.46
CAMK2B Q13554 1/20 0.46
CAMK2G Q13555 1/20 0.46
CAMK2D Q13557 1/20 0.46
CAMK2A Q9UQM7 1/20 0.46
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTR6 P50406 1/20 0.42
CA9 Q16790 2/20 0.41
CA12 O43570 1/20 0.41
TACR1 P25103 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
HTT P42858 1/20 0.40
GRIN1 Q05586 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316860 0.88 NQO1 (0.70) NQO1CDK4CCND1CCNE2CCNE1
SCHEMBL8316997 0.77 SIRT2 (0.53) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL8313203 0.70 NQO1 (1.00) NQO1CDK4CCND1CCNE2CCNE1
SCHEMBL8317087 0.70 ATM (0.58) ATMSMN1; SMN2CA9CA12CA1
SCHEMBL18669003 0.70 CA9 (0.61) ATMSMN1; SMN2CA9CA12CA1
SCHEMBL14708720 0.69 NQO1 (0.64) NQO1CDK4CCND1CCNE2CCNE1
SCHEMBL8318378 0.67 NQO1 (0.68) NQO1CDK4CCND1CCNE2CCNE1
SCHEMBL8195354 0.67 CDK4 (0.86) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL5769090 0.66 KCNN4 (0.51) ATMSMN1; SMN2CA9CA12CA1
SCHEMBL11099626 0.66 SMN1; SMN2 (0.58) ATMSMN1; SMN2CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP claimed