Cycloheptane

Cycloheptane

SCHEMBL8317003

C1CCCCCC1.O=C(O)NCC1CCc2ccccc2O1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.58
HTR1A P08908 3/20 0.49
HTR1D P28221 3/20 0.49
DRD2 P14416 5/20 0.48
DRD4 P21917 5/20 0.48
DRD3 P35462 5/20 0.48
DRD1 P21728 2/20 0.48
DRD5 P21918 2/20 0.48
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclopropane SCHEMBL6954169 1.00 CA2 (0.58) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL4935025 0.97 CA2 (0.60) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL23195321 0.86 CA2 (0.58) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL30152355 0.86 CA2 (0.58) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL1567983 0.86 CA2 (0.60) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL7319406 0.85 CA2 (0.54) CA2HTR1AHTR1D
SCHEMBL1380267 0.84 MTNR1A (0.62) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL1385775 0.84 MTNR1A (0.62) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL1380270 0.84 MTNR1A (0.62) CA2HTR1AHTR1DDRD2DRD4
SCHEMBL6955676 0.83 CA2 (0.58) CA2HTR1AHTR1DDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540914-B1 2-Aminomethylchromans as active ingredients in medicaments for the treatment of diseases of the central nervous system BAYER AG (DE) 1999-06-02 EP disclosed
EP-0540914-A1 2-Aminomethylchromans as active ingredients in medicaments for the treatment of diseases of the central nervous system BAYER AG (DE) 1993-05-12 EP disclosed