SCHEMBL8317093

SCHEMBL8317093

O=C1CCC(Nc2ncc3ncnc(Nc4cccc(Cl)c4)c3n2)CC1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.57
ERBB2 P04626 1/20 0.57
HPGD P15428 1/20 0.57
HTT P42858 1/20 0.57
CSNK2A2 P19784 1/20 0.53
CSNK2B P67870 1/20 0.53
CSNK2A1 P68400 1/20 0.53
FADS1 O60427 1/20 0.45
LCK P06239 1/20 0.44
BRAF P15056 1/20 0.43
CDK1 P06493 3/20 0.43
PRKCA P17252 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142831 0.92 EGFR (0.62) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8314630 0.88 EGFR (0.66) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319851 0.88 EGFR (0.64) EGFRERBB2HPGDHTT
SCHEMBL8801513 0.87 EGFR (0.62) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8316922 0.87 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8317806 0.87 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8460531 0.87 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8317294 0.87 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8317377 0.87 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A2
SCHEMBL8316918 0.87 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed