SCHEMBL8317294

SCHEMBL8317294

Clc1cccc(Nc2ncnc3cnc(NC4CCNCC4)nc23)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.58
ERBB2 P04626 1/20 0.58
HPGD P15428 1/20 0.58
HTT P42858 1/20 0.58
PAK4 O96013 1/20 0.54
CSNK2A1 P68400 3/20 0.51
CSNK2A2 P19784 1/20 0.51
CSNK2B P67870 1/20 0.51
FADS1 O60427 1/20 0.46
SYK P43405 1/20 0.45
LCK P06239 1/20 0.45
CYP1A2 P05177 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
MEN1 O00255 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142831 0.93 EGFR (0.62) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8316255 0.88 EGFR (0.67) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL7576672 0.88 EGFR (0.66) EGFRERBB2HPGDHTT
SCHEMBL8316922 0.88 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317806 0.88 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8460531 0.88 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8316918 0.88 EGFR (0.58) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317377 0.88 EGFR (0.58) EGFRERBB2HPGDHTTPAK4
SCHEMBL8317381 0.88 EGFR (0.58) EGFRERBB2HPGDHTTPAK4
SCHEMBL8317093 0.87 EGFR (0.57) EGFRERBB2HPGDHTTCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed