SCHEMBL8317141

SCHEMBL8317141

CC(C)(CO)Nc1ncc2ncnc(Nc3cccc(Cl)c3)c2n1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.53
FADS1 O60427 1/20 0.46
LCK P06239 1/20 0.46
FBP1 P09467 1/20 0.45
ERBB2 P04626 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316868 0.92 EGFR (0.53) EGFRFADS1LCKFBP1ERBB2
SCHEMBL8315733 0.89 EGFR (0.69) EGFRERBB2
SCHEMBL8316788 0.88 EGFR (0.58) EGFRFADS1LCKFBP1ERBB2
SCHEMBL8319419 0.88 EGFR (0.70) EGFR
SCHEMBL8318470 0.87 EGFR (0.48) EGFRERBB2
SCHEMBL8318372 0.86 EGFR (0.59) EGFRFBP1ERBB2
SCHEMBL8318939 0.85 EGFR (0.51) EGFRLCKFBP1ERBB2
SCHEMBL8313472 0.84 EGFR (0.53) EGFRFADS1LCKFBP1
SCHEMBL8315550 0.84 ABCG2 (0.51) EGFR
SCHEMBL8314176 0.81 EGFR (0.53) EGFRFADS1LCKERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed