SCHEMBL8315550

SCHEMBL8315550

CC(C)(CO)Nc1ncc2ncnc(Nc3cccc([N+](=O)[O-])c3)c2n1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.51
EGFR P00533 13/20 0.49
RAF1 P04049 1/20 0.45
BRAF P15056 1/20 0.45
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312686 0.93 ABCG2 (0.51) ABCG2EGFRRAF1BRAFMEN1
SCHEMBL8315105 0.89 ABCG2 (0.55) ABCG2EGFRRAF1BRAF
SCHEMBL8317827 0.85 ABCG2 (0.51) ABCG2EGFRRAF1BRAF
SCHEMBL8315733 0.84 EGFR (0.69) EGFR
SCHEMBL8317141 0.84 EGFR (0.53) EGFR
SCHEMBL8319419 0.84 EGFR (0.70) EGFR
SCHEMBL8316986 0.83 ABCG2 (0.53) ABCG2EGFRRAF1BRAF
SCHEMBL8313676 0.82 ABCG2 (0.53) ABCG2EGFRMEN1ALDH1A1MAPT
SCHEMBL8314074 0.82 ABCG2 (0.55) ABCG2EGFRRAF1BRAF
SCHEMBL8318939 0.81 EGFR (0.51) ABCG2EGFRRAF1BRAFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed