SCHEMBL8318939

SCHEMBL8318939

C#Cc1cccc(Nc2ncnc3cnc(NC(C)(C)CO)nc23)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.51
FBP1 P09467 2/20 0.48
GAK O14976 2/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
ERBB2 P04626 3/20 0.46
ERBB4 Q15303 2/20 0.46
PLK4 O00444 1/20 0.46
CIT O14578 1/20 0.46
AURKA O14965 1/20 0.46
EPHB6 O15197 1/20 0.46
SLC22A1 O15245 1/20 0.46
DAPK3 O43293 1/20 0.46
RIPK2 O43353 1/20 0.46
BUB1 O43683 1/20 0.46
KDM1A O60341 1/20 0.46
JAK2 O60674 1/20 0.46
RPS6KA4 O75676 1/20 0.46
STK17B O94768 1/20 0.46
STK10 O94804 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314305 0.93 EGFR (0.52) EGFRFBP1GAKALDH1A1MAPT
SCHEMBL8317979 0.89 EGFR (0.55) EGFRFBP1GAKALDH1A1MAPT
SCHEMBL8315733 0.86 EGFR (0.69) EGFRERBB2
SCHEMBL8319419 0.85 EGFR (0.70) EGFR
SCHEMBL8317141 0.85 EGFR (0.53) EGFRFBP1ERBB2LCK
SCHEMBL8317531 0.85 EGFR (0.51) EGFRFBP1GAKALDH1A1MAPT
SCHEMBL8316734 0.83 EGFR (0.55) EGFRFBP1GAKALDH1A1MAPT
SCHEMBL8316897 0.82 EGFR (0.50) EGFRFBP1GAKALDH1A1MAPT
SCHEMBL8315550 0.81 ABCG2 (0.51) EGFRALDH1A1MAPTRAF1BRAF
SCHEMBL8318849 0.81 EGFR (0.55) EGFRFBP1GAKALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed