SCHEMBL8317245

SCHEMBL8317245

Cc1cc(Cl)ccc1C(=O)Nc1cc(Cl)c(C(=O)N2CCc3cccn3-c3ccccc32)cc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 12/20 0.46
AVPR1A P37288 11/20 0.46
ALDH1A1 P00352 1/20 0.44
ABCB11 O95342 1/20 0.44
ADRB2 P07550 1/20 0.44
HTR1A P08908 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CHRM1 P11229 1/20 0.44
TBXA2R P21731 1/20 0.44
HTR2C P28335 1/20 0.44
HRH1 P35367 1/20 0.44
OPRM1 P35372 1/20 0.44
GLP1R P43220 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
FFAR4 Q5NUL3 1/20 0.44
GPR119 Q8TDV5 1/20 0.44
OXTR P30559 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315247 0.87 NPSR1 (0.44) AVPR2AVPR1AALDH1A1RAB9A
SCHEMBL8314766 0.85 AVPR2 (0.54) AVPR2AVPR1AOXTR
SCHEMBL7333870 0.83 AVPR2 (0.64) AVPR2AVPR1AALDH1A1OXTRNPC1
SCHEMBL8318107 0.81 AVPR2 (0.65) AVPR2AVPR1A
SCHEMBL7341288 0.78 AVPR2 (0.68) AVPR2AVPR1AOXTR
SCHEMBL8318709 0.78 AVPR2 (0.54) AVPR2AVPR1ANPC1RAB9A
SCHEMBL8312759 0.77 AVPR1A (0.55) AVPR2AVPR1A
SCHEMBL7337562 0.77 AVPR2 (0.44) AVPR2NPC1RAB9ASMN1; SMN2
SCHEMBL7334076 0.77 AVPR2 (0.68) AVPR2AVPR1AOXTRNPC1RAB9A
SCHEMBL7409772 0.76 AVPR2 (0.63) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed