SCHEMBL8317410

SCHEMBL8317410

Brc1cccc(Nc2ncnc3cnc(NCC4CCCO4)nc23)c1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.62
CSNK2A1 P68400 1/20 0.49
BRAF P15056 2/20 0.49
KCNH3 Q9ULD8 1/20 0.47
TNK2 Q07912 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319425 0.89 MAPT (0.56) EGFRCSNK2A1BRAFKCNH3
SCHEMBL8315088 0.89 EGFR (0.62) EGFRCSNK2A1BRAFKCNH3TNK2
SCHEMBL8316924 0.87 CSNK2A1 (0.65) EGFRCSNK2A1BRAFKCNH3
SCHEMBL8321243 0.85 MAPT (0.52) EGFRCSNK2A1BRAF
SCHEMBL8317434 0.84 EPHA2 (0.53) EGFRCSNK2A1BRAFTNK2
SCHEMBL8316693 0.82 EGFR (0.59) EGFRBRAFKCNH3TNK2
SCHEMBL6994869 0.79 MAPK1 (0.51) EGFRCSNK2A1BRAFKCNH3TNK2
SCHEMBL8316032 0.78 EGFR (0.72) EGFR
SCHEMBL8317824 0.78 EGFR (0.66) EGFR
SCHEMBL8315545 0.77 EGFR (0.72) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed