SCHEMBL8317434

SCHEMBL8317434

Clc1ccc(Nc2ncnc3cnc(NCC4CCCO4)nc23)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHA2 P29317 2/20 0.53
KDR P35968 2/20 0.53
BRAF P15056 2/20 0.49
TNK2 Q07912 10/20 0.48
EGFR P00533 2/20 0.48
HPGD P15428 2/20 0.48
ERBB2 P04626 1/20 0.48
HTT P42858 1/20 0.48
CHEK1 O14757 1/20 0.46
JAK2 O60674 1/20 0.46
ABL1 P00519 1/20 0.46
LCK P06239 1/20 0.46
ROS1 P08922 1/20 0.46
FGFR1 P11362 1/20 0.46
SRC P12931 1/20 0.46
TYK2 P29597 1/20 0.46
ALK Q9UM73 1/20 0.46
CSNK2A1 P68400 1/20 0.45
MEN1 O00255 2/20 0.45
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316693 0.92 EGFR (0.59) EPHA2KDRBRAFTNK2EGFR
SCHEMBL8319425 0.88 MAPT (0.56) BRAFEGFRHPGDHTTCSNK2A1
SCHEMBL8317410 0.84 EGFR (0.62) BRAFTNK2EGFRCSNK2A1
SCHEMBL8315088 0.84 EGFR (0.62) BRAFTNK2EGFRHPGDCSNK2A1
SCHEMBL8316924 0.82 CSNK2A1 (0.65) BRAFEGFRCSNK2A1LMNAKMT2A
SCHEMBL8321243 0.81 MAPT (0.52) BRAFEGFRHTTCSNK2A1LMNA
SCHEMBL6994869 0.80 MAPK1 (0.51) BRAFTNK2EGFRERBB2HTT
SCHEMBL8316240 0.78 EGFR (0.69) EPHA2KDRBRAFEGFRHPGD
SCHEMBL8314200 0.78 EGFR (0.64) BRAFEGFRHPGDERBB2HTT
SCHEMBL8317784 0.76 EGFR (0.49) EGFRHPGDERBB2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed