SCHEMBL8317520

SCHEMBL8317520

CN1CCC(Nc2ncc3ncnc(Nc4cccc([N+](=O)[O-])c4)c3n2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.63
ERBB2 P04626 1/20 0.63
HPGD P15428 1/20 0.63
HTT P42858 1/20 0.63
BRD4 O60885 2/20 0.50
BRAF P15056 2/20 0.49
ABCG2 Q9UNQ0 2/20 0.48
PKM P14618 1/20 0.47
FLT3 P36888 1/20 0.45
TYRO3 Q06418 1/20 0.45
MERTK Q12866 1/20 0.45
GAS6 Q14393 1/20 0.45
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
EIF2AK2 P19525 1/20 0.44
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CDK5 Q00535 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315091 0.92 ABCG2 (0.54) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313619 0.88 GSK3A (0.56) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313626 0.88 GSK3A (0.56) EGFRERBB2HPGDHTTBRAF
SCHEMBL8317605 0.88 ABCG2 (0.50) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313945 0.88 GSK3A (0.56) EGFRERBB2HPGDHTTBRAF
SCHEMBL8317920 0.88 EGFR (0.51) EGFRERBB2HPGDHTTBRAF
SCHEMBL8316755 0.88 CTSL (0.57) EGFRERBB2HPGDHTTABCG2
SCHEMBL8318742 0.88 ABCG2 (0.50) EGFRERBB2HPGDHTTABCG2
SCHEMBL8317918 0.88 EGFR (0.51) EGFRERBB2HPGDHTTBRAF
SCHEMBL8313514 0.87 ABCG2 (0.48) EGFRERBB2HPGDHTTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed