SCHEMBL8317624

SCHEMBL8317624

C=C1CC(C(C#N)c2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
TRPA1 O75762 1/20 0.39
TSHR P16473 1/20 0.39
SLC6A3 Q01959 2/20 0.36
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
IDO1 P14902 2/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7355279 0.80 CHRNB4 (0.53) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL961750 0.77 SLC6A3 (0.53) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL961019 0.77 SLC6A3 (0.57) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL13124077 0.76 SLC6A3 (0.58) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL959762 0.76 SLC6A3 (0.58) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL8317202 0.74 CHRNB4 (0.44) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL8191324 0.73 CHRNB4 (0.46) CHRNB4CHRNA3SLC6A3SLC6A2SLC6A4
SCHEMBL8319051 0.73 CHRNB4 (0.43) CHRNB4CHRNA3TRPA1TSHRSLC6A3
SCHEMBL493477 0.73 CHRNB4 (0.46) CHRNB4CHRNA3TRPA1TSHRSLC6A3
Hydrochloric Acid SCHEMBL2586181 0.71 CHRNB4 (0.45) CHRNB4CHRNA3SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923536-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION Pharmacia & Upjohn Aktiebolag (SE) 1999-06-23 EP disclosed
WO-1998004517-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-02-05 WO disclosed