SCHEMBL8317897

SCHEMBL8317897

CCOC(=O)c1ccc(NC(=O)c2cccc(C(F)(F)F)c2)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.57
CYP1A2 P05177 2/20 0.54
RAB9A P51151 2/20 0.54
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
LMNA P02545 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
MAPT P10636 1/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
PTGS1 P23219 2/20 0.51
HTT P42858 1/20 0.51
TAS1R3 Q7RTX0 1/20 0.51
TAS1R1 Q7RTX1 1/20 0.51
TAS1R2 Q8TE23 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27532598 0.83 MEN1 (0.59) GAACYP1A2RAB9AALDH1A1CYP3A4
SCHEMBL8313664 0.83 CYP1A2 (0.50) GAACYP1A2RAB9AALDH1A1KDM4E
SCHEMBL8313189 0.83 TRPV1 (0.50) GAACYP1A2RAB9AALDH1A1KDM4E
SCHEMBL28007500 0.82 RAB9A (0.70) RAB9AALDH1A1LMNAMAPTMEN1
SCHEMBL30786693 0.82 CES2 (0.61) ALDH1A1LMNANPSR1MAPTMEN1
SCHEMBL1994068 0.82 CES2 (0.61) ALDH1A1LMNANPSR1MAPTMEN1
SCHEMBL8315698 0.81 RAB9A (0.53) GAACYP1A2RAB9AALDH1A1KDM4E
SCHEMBL8314651 0.81 RAB9A (0.47) GAACYP1A2RAB9AALDH1A1KDM4E
SCHEMBL8816442 0.81 RAB9A (0.62) GAACYP1A2RAB9AALDH1A1KDM4E
SCHEMBL8311983 0.80 RAB9A (0.58) GAACYP1A2RAB9AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed
CN-1106812-A Tricyclic diaza * vasopressin antagonists and oxytocin antagonists AMERICAN CYANAMID CO (US) 1995-08-16 CN disclosed