SCHEMBL8317898

SCHEMBL8317898

CC(C)N(C)c1c(N)cccc1F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.34
CYP3A4 P08684 2/20 0.33
TSHR P16473 2/20 0.33
PIK3CA P42336 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
TAAR1 Q96RJ0 1/20 0.32
CD44 P16070 1/20 0.30
ALDH1A1 P00352 2/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
KDM4E B2RXH2 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27010079 0.86 TAAR1 (0.38) AOC3DRD2DRD3TDP1TAAR1
SCHEMBL26122242 0.74 CYP19A1 (0.35) CYP3A4TSHRPIK3CATDP1ALDH1A1
SCHEMBL8313252 0.70 TDP1 (0.43) TSHRTDP1ALDH1A1HSD17B10SMN1; SMN2
SCHEMBL24316013 0.68 TAAR1 (0.34) AOC3DRD2DRD3TDP1TAAR1
SCHEMBL30936694 0.67 BRD4 (0.36) TDP1
SCHEMBL30936652 0.67 PABPC1 (0.37) CYP3A4ALDH1A1KDM4ESMN1; SMN2
SCHEMBL9607569 0.67 CYP3A4 (0.39) CYP3A4TSHRPIK3CATDP1CD44
SCHEMBL27010080 0.67 TAAR1 (0.41) AOC3TDP1TAAR1ALDH1A1HPGD
SCHEMBL23278085 0.67 CHEK1 (0.42) AOC3CYP3A4TSHRPIK3CATDP1
SCHEMBL7697624 0.67 KCNH2 (0.42) AOC3TSHRTDP1TAAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929072-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY LIMITED (GB) 1999-07-27 US disclosed
WO-1999010346-A1 BENZOTHIADIAZINYL-INDOLE DERIVATIVES AND THEIR USE AS SEROTONIN RECEPTOR LIGANDS ELI LILLY AND COMPANY LIMITED (GB) 1999-03-04 WO disclosed
EP-0897921-A1 Benzothiadiazinyl-indole derivatives and their use as serotonin receptor ligands ELI LILLY AND COMPANY LIMITED (GB) 1999-02-24 EP disclosed