SCHEMBL8318072

SCHEMBL8318072

Cc1cccc(Nc2ncnc3cnc(NC4CCCC4)nc23)c1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.71
ERBB2 P04626 1/20 0.55
HPGD P15428 1/20 0.55
HTT P42858 1/20 0.55
MAPK3 P27361 4/20 0.50
MAPK1 P28482 4/20 0.50
SYK P43405 4/20 0.50
KCNH2 Q12809 4/20 0.50
AURKB Q96GD4 4/20 0.50
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ADORA1 P30542 1/20 0.49
BRAF P15056 1/20 0.48
GP6 Q9HCN6 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319537 0.99 EGFR (0.69) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8318282 0.98 EGFR (0.71) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8319428 0.96 EGFR (0.73) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8319108 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8313632 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8317834 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8319114 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8313624 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8316255 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3
SCHEMBL8322339 0.91 EGFR (0.67) EGFRERBB2HPGDHTTMAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed