SCHEMBL8322339

SCHEMBL8322339

Cc1cccc(Nc2ncnc3cnc(N[C@H]4CC[C@H](O)CC4)nc23)c1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.67
BRAF P15056 1/20 0.59
ERBB2 P04626 1/20 0.53
HPGD P15428 1/20 0.53
HTT P42858 1/20 0.53
SYK P43405 4/20 0.48
KCNH2 Q12809 4/20 0.48
MAPK3 P27361 2/20 0.47
MAPK1 P28482 2/20 0.47
AURKB Q96GD4 2/20 0.47
JUN P05412 1/20 0.47
MAPK10 P53779 1/20 0.47
MAPK8 P45983 1/20 0.47
MAPK9 P45984 1/20 0.47
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319114 1.00 EGFR (0.67) EGFRBRAFERBB2HPGDHTT
SCHEMBL8319108 1.00 EGFR (0.67) EGFRBRAFERBB2HPGDHTT
SCHEMBL8319428 0.95 EGFR (0.73) EGFRBRAFERBB2HPGDHTT
SCHEMBL8318282 0.91 EGFR (0.71) EGFRBRAFERBB2HPGDHTT
SCHEMBL8318072 0.91 EGFR (0.71) EGFRBRAFERBB2HPGDHTT
SCHEMBL8313624 0.90 EGFR (0.67) EGFRBRAFERBB2HPGDHTT
SCHEMBL8313632 0.90 EGFR (0.67) EGFRBRAFERBB2HPGDHTT
SCHEMBL8319537 0.90 EGFR (0.69) EGFRBRAFERBB2HPGDHTT
SCHEMBL8318922 0.89 EGFR (0.62) EGFRBRAFERBB2HPGDHTT
SCHEMBL8318928 0.89 EGFR (0.62) EGFRBRAFERBB2HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed