SCHEMBL8318535

SCHEMBL8318535

COC(=O)c1cc2c(C)ccc(Cl)c2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
XDH P47989 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CYP1A2 P05177 1/20 0.41
NR4A2 P43354 2/20 0.41
ALPL P05186 2/20 0.41
ABL1 P00519 4/20 0.40
SRC P12931 4/20 0.40
LMNA P02545 1/20 0.38
PTGS2 P35354 1/20 0.38
ULK1 O75385 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.38
FBP1 P09467 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319918 0.89 GLA (0.48) GLAGAAXDHCDK1CCNB1
SCHEMBL8320394 0.88 GLA (0.45) GLAGAAXDHCDK1CCNB1
SCHEMBL8318563 0.87 GLA (0.49) GLAGAAXDHCYP1A2NR4A2
SCHEMBL24020849 0.85 IDO1 (0.46) GLAGAAXDHCDK1CCNB1
SCHEMBL8322794 0.84 KDM4E (0.57) GLAGAAXDHCDK1CCNB1
SCHEMBL30184708 0.84 XDH (0.50) GLAGAAXDHCDK1CCNB1
SCHEMBL10093729 0.83 GLA (0.46) GLAGAAXDHCYP1A2LMNA
SCHEMBL19014158 0.82 IDO1 (0.49) GLAGAAXDHCYP1A2ALPL
SCHEMBL8319614 0.82 GAA (0.62) GLAGAAXDHCYP1A2LMNA
SCHEMBL23049740 0.79 XDH (0.44) GLAGAAXDHCDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-9048755-A None JP disclosed
WO-2017106352-A1 CAFFEINE INHIBITORS OF MTHFD2 AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-06-22 WO disclosed
US-5866594-A Indole-2-carboxylate derivatives and fungicidal compositions for agricultural or horticultural use containing the derivatives as active component OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1999-02-02 US disclosed
EP-0791582-A1 INDOLE-2-CARBOXYLIC ESTER DERIVATIVES AND AGRICULTURAL AND HORTICULTURAL BACTERIOCIDES CONTAINING THE SAME AS THE ACTIVE INGREDIENT OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1997-08-27 EP disclosed
JP-H0948755-A INDOLE-2-CARBOXYLIC ACID ESTER DERIVATIVE OTSUKA CHEM CO LTD 1997-02-18 JP disclosed