SCHEMBL8318539

SCHEMBL8318539

Clc1ccc2c(c1)OC[C@H]1CN(Cc3ccccc3)C[C@H]21

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.81
DRD3 P35462 13/20 0.81
DPP4 P27487 1/20 0.55
SIGMAR1 Q99720 1/20 0.44
CCR5 P51681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8903147 0.99 DRD2 (0.80) DRD2DRD3DPP4SIGMAR1CCR5
Hydrochloric Acid SCHEMBL8685262 0.99 DRD2 (0.80) DRD2DRD3DPP4SIGMAR1CCR5
SCHEMBL32660192 0.90 DRD2 (0.67) DRD2DRD3DPP4SIGMAR1CCR5
SCHEMBL8318315 0.90 DRD2 (1.00) DRD2DRD3DPP4
SCHEMBL8313033 0.90 DRD2 (1.00) DRD2DRD3DPP4
Hydrochloric Acid SCHEMBL8685090 0.89 DRD2 (0.97) DRD2DRD3DPP4
Hydrochloric Acid SCHEMBL8686313 0.89 DRD2 (0.97) DRD2DRD3DPP4
Hydrochloric Acid SCHEMBL8902652 0.89 DRD2 (0.97) DRD2DRD3DPP4
SCHEMBL8317999 0.85 DRD2 (1.00) DRD2DRD3SIGMAR1
SCHEMBL29960315 0.85 DRD2 (1.00) DRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691342-B1 Benzopyran derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1999-04-28 EP disclosed
EP-0691342-A1 Benzopyrane derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed