SCHEMBL8319612

SCHEMBL8319612

COc1cccc(/C(=C(\N)C#N)c2cc(OC)cc(OC)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.58
PRSS1 P07477 1/20 0.54
PRSS2 P07478 1/20 0.54
PRSS3 P35030 1/20 0.54
PDE4A P27815 3/20 0.54
PDE4B Q07343 3/20 0.54
PDE4C Q08493 3/20 0.54
PDE4D Q08499 3/20 0.54
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
NPC1 O15118 7/20 0.49
RAB9A P51151 5/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
PKM P14618 1/20 0.49
XBP1 P17861 1/20 0.49
MAPK1 P28482 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
STS P08842 2/20 0.46
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8269327 1.00 PARP1 (0.58) PARP1PRSS1PRSS2PRSS3PDE4A
SCHEMBL4816445 0.84 PDE4A (0.56) PARP1PRSS1PRSS2PRSS3PDE4A
SCHEMBL8269336 0.83 PARP1 (0.66) PARP1PRSS1PRSS2PRSS3PDE4A
SCHEMBL17122434 0.81 PARP1 (0.57) PARP1PRSS1PRSS2PRSS3PDE4A
SCHEMBL10897886 0.75 CES2 (0.67) PARP1PRSS1PRSS2PRSS3PDE4A
SCHEMBL29503138 0.74 PARP1 (1.00) PARP1PRSS1PRSS2PRSS3CES2
SCHEMBL283787 0.74 PARP1 (1.00) PARP1PRSS1PRSS2PRSS3CES2
Hydrochloric Acid SCHEMBL407554 0.73 PARP1 (0.96) PARP1PRSS1PRSS2PRSS3CES2
SCHEMBL4820908 0.73 CES2 (0.69) PARP1PRSS1PRSS2PRSS3PDE4A
Hydrochloric Acid SCHEMBL4377519 0.73 PARP1 (0.96) PARP1PRSS1PRSS2PRSS3CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078144-A2 DIPHENYLETHYLENE COMPOUNDS AND USES THEREOF CELGENE CORPORATION (US) 2004-09-16 WO disclosed