SCHEMBL8319689

SCHEMBL8319689

O=C(C[CH]NC(=O)OCc1ccccc1)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
MAPK1 P28482 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 2/20 0.51
POLB P06746 2/20 0.51
RAB9A P51151 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
LMNA P02545 1/20 0.50
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
GAA P10253 1/20 0.48
HTT P42858 1/20 0.48
MIF P14174 1/20 0.47
HCAR2 Q8TDS4 1/20 0.46
SLC6A2 P23975 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10556498 0.89 HTT (0.53) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL7709972 0.86 SYK (0.50) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL8322922 0.84 ALDH1A1 (0.51) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL4291030 0.83 ALDH1A1 (0.54) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL1415895 0.83 ALDH1A1 (0.55) ALDH1A1L3MBTL1SMN1; SMN2NPC1POLB
SCHEMBL8318380 0.81 SMN1; SMN2 (0.54) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL28661503 0.81 SMN1; SMN2 (0.58) ALDH1A1L3MBTL1SMN1; SMN2NPC1POLB
SCHEMBL8775648 0.80 ALDH1A1 (0.56) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL8546866 0.79 HTT (0.57) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL3725206 0.79 ALDH1A1 (0.50) ALDH1A1L3MBTL1SMN1; SMN2NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994342-A 3-(substituted methyl)-4-oxa-1-azabicyclo[3.2.0]heptan-7-one derivatives useful as antitumor agents TAIHO PHARMACEUTICAL CO., LTD. (JP) 1999-11-30 US disclosed
EP-0688324-A1 NOVEL 3-(SUBSTITUTED METHYL)-4-OXA-1-AZABICYCLO 3.2.0]HEPTAN-7-ONE DERIVATIVES USEFUL AS ANTITUMOR AGENTS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1995-12-27 EP disclosed
WO-1995018807-A1 NOVEL 3-(SUBSTITUTED METHYL)-4-OXA-1-AZABICYCLO[3.2.0]HEPTAN-7-ONE DERIVATIVES USEFUL AS ANTITUMOR AGENTS TAIHO PHARMACEUTICAL CO. LIMITED (JP) 1995-07-13 WO disclosed