SCHEMBL8319699

SCHEMBL8319699

CCCc1c(C#N)cnc2nc(N)nc(N)c12

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
DHFR P00374 10/20 0.38
SLC2A1 P11166 1/20 0.36
CSNK1A1 P48729 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323430 0.92 KDM4E (0.42) KDM4EMEN1GAATSHRHTT
SCHEMBL9067611 0.80 TP53 (0.43) DHFRSLC2A1CSNK1A1CLK4
SCHEMBL4222830 0.78 DHFR (0.47) DHFRSLC2A1CSNK1A1CLK4
SCHEMBL8322368 0.76 DHFR (0.46) DHFRSLC2A1
SCHEMBL8468661 0.76 DHFR (0.43) DHFRSLC2A1
SCHEMBL8324477 0.75 DHFR (0.41) DHFRSLC2A1
SCHEMBL8320187 0.73 MAPK1 (0.42) KDM4EMEN1GAATSHRHTT
SCHEMBL20641250 0.68 CSNK1A1 (0.51) KDM4EMEN1GAATSHRHTT
SCHEMBL20641252 0.68 HSP90AA1 (0.47) KDM4EMEN1GAATSHRHTT
SCHEMBL26324937 0.67 KDM5A (0.43) KDM4EMEN1GAATSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0638079-B1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION STANFORD RES INST INT (US) 1999-12-15 EP disclosed
US-5536724-A Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins SRI INTERNATIONAL (US) 1996-07-16 US disclosed
EP-0638079-A1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1995-02-15 EP disclosed
WO-1993022312-A1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1993-11-11 WO disclosed