SCHEMBL8319798

SCHEMBL8319798

O=C=C(c1ccccc1)c1ccncc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.59
MEN1 O00255 1/20 0.59
ALDH1A1 P00352 3/20 0.53
CYP1A2 P05177 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP2C9 P11712 2/20 0.53
HPGD P15428 2/20 0.53
CYP2C19 P33261 2/20 0.53
PLOD2 O00469 1/20 0.53
PLOD3 O60568 1/20 0.53
PLOD1 Q02809 1/20 0.53
HIF1A Q16665 1/20 0.53
NAPRT Q6XQN6 1/20 0.48
HTT P42858 1/20 0.46
JAK2 O60674 1/20 0.46
TYK2 P29597 1/20 0.46
KCNK3 O14649 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP19A1 P11511 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL80355 0.86 CES1 (0.48) KMT2AMEN1ALDH1A1CYP3A4HPGD
SCHEMBL28632577 0.84 CES1 (0.46) KMT2AMEN1ALDH1A1CYP3A4HPGD
SCHEMBL229650 0.75 KMT2A (1.00) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL3074392 0.75 KMT2A (0.74) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL25983244 0.74 KMT2A (0.65) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL733007 0.74 KMT2A (0.65) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL18983076 0.74 KMT2A (0.65) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL17728703 0.74 KMT2A (0.58) KMT2AALDH1A1NAPRTKCNK3L3MBTL1
Benzamide SCHEMBL28787993 0.71 CYP3A4 (0.73) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL17115264 0.70 KMT2A (0.60) KMT2AMEN1ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871444-A4 2,5-SUBSTITUTED ARYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO INC (US) 1999-01-13 EP disclosed
EP-0871444-A1 2,5-SUBSTITUTED ARYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE Merck & Co., Inc. (US) 1998-10-21 EP disclosed